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Products > GPCR > Opioid receptor > ADL 5859
Product name : ADL 5859
Item : cc30
Price : 200mg, $1250;500mg, $2090; 1g $2995; 2g, $4395
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239.
CAS : 850173-95-4
Molecular Weight : 428.95
Formula : C₂₄H₂₉ClN₂O₃
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Details:
ADL5859 is an δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM). Preclinical work suggests that δ-specific agonists may exhibit superior analgesic properties to µ agonists whilst avoiding some of their common and undesirable side-effects. ADL-5859 is an agonist agent that selectively stimulates the δ-opioid receptor with potential application in a wide range of inflammatory, neuropathic and acute pain conditions. [1][2]
 
Reference:
[1] J Med. Chem. 2008, 51, 5893-5896.
[2] J Pharmacol. Exp. Ther. 2012, 342, 799-807.
 
 
Chemical Information
Molecular Weight (WM):
428.95
Formula:
C24H28N2O3.HCl
CAS No:
850173-95-4, 850305-06-5 (free base)
Purity:
≥ 98%
Synonyms:
ADL 5859
 
DMSO ≥ 86 mg/mL
Solubility (25℃)
Water ≥ 11 mg/mL
 
Ethanol < 1 mg/mL
 
2 years     -20℃        Powder
Stability:
2 weeks     -4℃        in DMSO
 
2 months    -80℃       in DMSO
 
Quality control data:
Quality control by 1H-NMR, 13C-NMR, HPLC and LCMS.
Product will be shipped with supporting analytical data.
 
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
 
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE.

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