Product name : Clobenpropit (VUF 9153)
Item : cc780
Price : 200mg, $950;500mg, $1695; 1g, $2490; 2g, $3590
contact : Send inquiry to: info@acesobio.com,or by fax to: 1-845-673-1239
CAS : 145231-45-4
Molecular Weight : 470.65
Formula : C14H17ClN4S 2HBr
Storage : at -20°C
Additional information : We offer significant discount for bulky quantity order
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Clobenpropit (VUF-9153) has been shown to be an extremely potent (pA2 = 9.93) and selective histamine H3 receptor antagonist. This compound has been found to enhance the release of GABA, which protects against NMDA-induced exitotoxicity. Further experiments suggest that clobenpropit dihydrobromide my inhibit the binding of iodophenpropit, and therefor may possess the ability to cross the blood-brain barrier. [1][2]
Reference:
[1] Eur. J Pharmacol. 1994, 260, 23-28.
[2] Eur. J Pharmacol. 2007, 563, 117-123.
Chemical Information
PLEASE KEEP THE PRODUCT UNDER -20℃ FOR LONG-TERM STORAGE.
NOT FOR HUMAN OR VETERINARY DIAGNOSTIC OR THERAPEUTIC USE. |
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